Document Type

Article

Publication Date

5-16-2024

Keywords

JGM, RNA Splicing Factors, Humans, Animals, Phosphoproteins, Mutation, Hematologic Neoplasms, Mice, RNA Splicing, DEAD-box RNA Helicases, Hematopoiesis, HEK293 Cells, Introns, RNA Helicases, RNA-Binding Proteins

JAX Source

Mol Cell. 2024;84(10):1886-903.e10.

ISSN

1097-4164

PMID

38688280

DOI

https://doi.org/10.1016/j.molcel.2024.04.006

Abstract

Mutations in the RNA splicing factor gene SF3B1 are common across hematologic and solid cancers and result in widespread alterations in splicing, yet there is currently no therapeutic means to correct this mis-splicing. Here, we utilize synthetic introns uniquely responsive to mutant SF3B1 to identify trans factors required for aberrant mutant SF3B1 splicing activity. This revealed the G-patch domain-containing protein GPATCH8 as required for mutant SF3B1-induced splicing alterations and impaired hematopoiesis. GPATCH8 is involved in quality control of branchpoint selection, interacts with the RNA helicase DHX15, and functionally opposes SURP and G-patch domain containing 1 (SUGP1), a G-patch protein recently implicated in SF3B1-mutant diseases. Silencing of GPATCH8 corrected one-third of mutant SF3B1-dependent splicing defects and was sufficient to improve dysfunctional hematopoiesis in SF3B1-mutant mice and primary human progenitors. These data identify GPATCH8 as a novel splicing factor required for mis-splicing by mutant SF3B1 and highlight the therapeutic impact of correcting aberrant splicing in SF3B1-mutant cancers.

Creative Commons License

Creative Commons Attribution 4.0 International License
This work is licensed under a Creative Commons Attribution 4.0 International License.

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